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Pharmaceutical Research Division, Takeda Chemical Industries, Ltd. | 論文
- STRUCTURES AND ACTIVITIES OF TANNINS IN CRUDE DRUGS (3)
- Characterization of the CYP2C8 Active Site by Homology Modeling
- Characterization of the CYP3A4 Active Site by Homology Modeling
- Orally Active CCR5 Antagonists as Anti-HIV-1 Agents : Synthesis and Biological Activity of 1-Benzothiepine 1, 1-Dioxide and 1-Benzazepine Derivatives Containing a Tertiary Amine Moiety
- Kinetic Resolutions of Indan Derivatives Using Bacteria(Microbiology & Fermentation Technology)
- Orally Active CCR5 Antagonists as Anti-HIV-1 Agents 2 : Synthesis and Biological Activities of Anilide Derivatives Containing a Pyridine N-Oxide Moiety
- CCR5 Antagonists as Anti-HIV-1 Agents.1. Synthesis and Biological Evaluation of 5-Oxopyrrolidine-3-carboxamide Derivatives
- Constituents of Geranium thunbergii SIEB. et ZUCC. XV. Modified Dehydroellagitannins, Geraniinic Acids B and C, and Phyllanthusiin F
- In vitro antimicrobial activity of T-91825, a novel anti-MRSA cephalosporin, and in vivo anti-MRSA activity of its prodrug, TAK-599
- Studies on Anti-MRSA Parenteral Cephalosporins : IV. A Novel Water-soluble N-Phosphono Type Prodrug for Parenteral Administration
- Studies on Anti-MRSA Parenteral Cephalosporins : III. Synthesis and Antibacterial Activity of 7β-[2-(5-Amino-1,2,4-thiadiazol-3-yl)-2(Z)-alkoxyiminoacetamido]-3-[(E)-2-(1-alkylimidazo[1,2-b]pyridazinium-6-yl)thiovinyl]-3-cephem-4-carboxylates and Related
- Studies on Anti-MRSA Parenteral Cephalosporins : II. Synthesis and Antibacterial Activity of 7β-[2-(5-Amino-1,2,4-thiadiazol-3-yl)-2(Z)-alkoxyiminoacetamido]-3-(substituted imidazo[1,2-b]pyridazinium-1-yI)methyl-3-cephem-4-carboxylates and Related Compoun
- Studies on Anti-MRSA Parenteral Cephalosporins : I. Synthesis and Antibacterial Activity of 7β-[2-(5-Amino-1,2,4-thiadiazol-3-yl)-2(Z)-hydroxyiminoacetamido]-3-(substituted imidazo[1,2-b]-pyridazinium-1-yl)methyl-3-cephem-4-carboxylates and Related Compou
- Synthetic Studies on Condensed-Azole Derivatives. V. Synthesis and Anti-asthmatic Activities of ω-Sulfamoylalkyloxy[1,2,4]triazolo[1,5-b]-pyridazines
- Synthetic Studies on Condensed-Azole Derivatives. IV. Synthesis and Anti-asthmatic Activities of ω-Sulfamoylalkyloxyimidazo[1,2-b]pyridazines
- The First Example for Cycloenantiomeric Hexahomooxacalix[3]arenes
- Optically Active Antifungal Azoles. IV. Synthesis and Antifungal Activity of (2R, 3R)-3-Azolyl-2-(substituted phenyl)-1-(1H-1,2,4-triazol-1-yl)-2-butanols
- Optically Active Antifungal Azoles. II. Synthesis and Antifungal Activity of Polysulfide Derivatives of (2R, 3R)-2-(2,4-Difluorophenyl)-3-mercapto-1-(1H-1,2,4-triazol-1-yl)-2-butanol
- EG-VEGF/Prokineticins Are Cognate Ligands for Two Closely Related Orphan G-Protein-Coupled Receptors
- Pyloricidins, Novel Anti-Helicobacter pylori Antibiotics Produced by Bacillus sp. : II. Isolation and Structure Elucidation
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