ニトロフラン誘導体の研究(第6報) : 2-(5-Nitro-2-furyl)vinylpyridinemethanol類, および2-(5-Nitro-2-furyl)vinylpyridine carboxylic acid類の合成
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In order to examine their antibacterial activity, hydroxymethyl- or acetoxymethyl-2-[2-(5-nitro-2-furyl)vinyl]pyridines (I) and their N-oxides (I'), and 2-[2-(5-nitro-2-furyl)vinyl]-pyridinecarboxylic acids (II) were synthesized. For the synthesis of 6- or 4-hydroxymethyl- or -acetoxymethyl-2-[2-(5-nitro-2-furyl)-vinyl]pyridines (Ia, b, e, f), rearrangement of the N-oxide group in 6-methyl-2-[2-(5-nitro-2-furyl)vinyl]-pyridine 1-oxide in acetic anhydride was attempted and the objective Ia, Ib, Ie, and If were obtained, accompanied by the byproduct formation of a pyridinol derivative, in which oxygen in N-oxide group had undergone rearrangement to the pyridine ring.
- 公益社団法人日本薬学会の論文
- 1966-11-25
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