Condensed Thienopyrimidines. IV. : Synthesis and Gastric Antisecretory Activity of 2,3-Dihydro-5H-oxazolothienopyrimidine Derivatives

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概要

• 論文の詳細を見る

• 2,3-Dihydro-5H-oxazolo[3,2-a]thieno[3,2-d]-(2a-d), [3,4-d]-(2e-h), and [2,3-d]pyrimidine derivatives (2i, j) were synthesized and evaluated for gastric antisecretory activity. These analogues (2) were prepared stepwise starting from formylthiophenecarbamates (4). The structure-activity relationships of these compounds are discussed.

• 公益社団法人日本薬学会の論文
• 1989-10-25

著者

• 田端 敬一

  三共(株)ライセンス部

• 杉山 充男

  Medicinal Chemistry Research Laboratories

• 坂本 俊明

  Medicinal Chemistry Research Laboratories

• 田端 敬一

  Biological Research Laboratories

• 福見 宏

  Medicinal Chemistry Research Laboratories, Sankyo Co., Ltd.,

• 福見 宏

  Medicinal Chemistry Research Laboratories Sankyo Co. Ltd.

• 坂本 俊明

  Medicinal Chemistry Research Laboratories Sankyo Co. Ltd.

• 杉山 充男

  Medicinal Chemistry Research Laboratories Sankyo Co. Ltd.

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