A novel preparation of 3-hydroxy-3H-indole-3-ethanamines and -3H-indole-3-acetamides having either a 4-morpholinyl or 1-pyrrolidinyl group at the 2-position
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概要
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A novel synthetic method is discovered for 3-hydroxy-3H-indole-3-ethanamines and -3H-indole-3-acetamides having either a 4-morpholinyl or 1-pyrrolidinyl group at the 2-position by reacting the corresponding 1-hydroxyindoles with enamines in the presence of tosyl or mesyl chloride. A plausible mechanism is proposed.
- 日本複素環化学研究所の論文
- 2004-01-01
日本複素環化学研究所 | 論文
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