10-Aryl-3,3-dimethyl-2,3,4,10-tetrahydro-1H-pyrrolo[3,4-c][1,5]benzothiazepin-1-oneの合成
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概要
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3-Arylmethylene-5,5-dimethyltetramic acids (5a-i) were synthesized from 5,5-dimethyltetramic acid (3) and aromatic aldehydes by an acid catalyzed aldol condensation. 10-Aryl-3,3-dimethyl-2,3,4,10-tetrahydro-1H-pyrrolo [3,4-c] [1,5] benzothiazepin-1-ones (9a-g) were prepared by Michael reaction between 2-aminobenzenethiol and 3-arylmethylene-5,5-dimethyltetramic acids in good yield.
- 公益社団法人日本薬学会の論文
- 1984-09-25
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