Polyoxin Analogs. I. Synthesis of Aminoacyl Derivatives of 5'-Amino-5'-deoxyuridine

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概要

• 論文の詳細を見る

• 5'-δ-Carbamoyloxy-L-x-aminovaleramido-5'-deoxyuridine, a polyoxin analog, was prepared by the reaction of 5'-amino-5'-deoxy-2', 3'-O-isopropylideneuridine and N-carbobenzoxy-L-α-aminovalero-δ-lactone, followed by carbamoylation and the removal of the protective groups. Several other ω-substituted aminoacyl derivatives were also prepared utilizing the activated ester method and the mixed anhydride method. All these compounds showed no polyoxin-activity.

• 公益社団法人日本薬学会の論文
• 1971-03-25

著者

• 磯野 清

  The Institute Of Physical And Chemical Research

• 鈴木 三郎

  The Institute Of Physical And Chemical Research

• 東 常政

  The Institute of Physical and Chemical Research

• 東 常政

  The Institute Of Physical And Chemical Research:(present Address)research Division Kaken Chemical Co

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• Transnucleosidation : An Improved Method for Transglycosylation from Pyrimidines to Purines
• Polyoxin Analogs. III. Synthesis and Biological Activity of Aminoacyl Derivatives of Polyoxins C and L
• Formation and Characterization of 5'-Deoxy-5', 6-epimino-5,6-dihydro-2', 3'-O-isopropylideneuridine
• Polyoxin Analogs. I. Synthesis of Aminoacyl Derivatives of 5'-Amino-5'-deoxyuridine
• 37 ポリオキシンの構造研究

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