A Versatile Synthesis of 1-Aryl-2-nitro-3-(3,4-, 5-trimethoxyphenyl)-propenes as Precursors of Novel Mescaline Derivatives

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概要

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• A convenient one-step procedure to synthesize the title compounds (3a-v) by the reaction between 1,2,3-trimethoxy-5-(2-nitroethyl)benzene (1) and aromatic or heterocyclic aldehydes is reported. The obtained 1-aryl-2-nitro-3-(3,4,5-trimethoxyphenyl)propenes can easily be reduced to provide new mescaline derivatives. As an example, 1-(3-indolyl)-2-amino-3-(3,4,5-trimethoxyphenyl)propane (4), which contains in the same molecule the structural features of both mescaline and tryptamine, has been prepared.

• 公益社団法人日本薬学会の論文
• 1986-04-25

著者

• Royer Rene

  Service De Chimie De L'institut Curie E.r. N°213 Cnrs

• Dauzonne Daniel

  Service De Chimie De L'institut Curie E.r. N° 213 Cnrs

関連論文

• A Versatile Synthesis of 1-Aryl-2-nitro-3-(3,4-, 5-trimethoxyphenyl)-propenes as Precursors of Novel Mescaline Derivatives

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