A Facile Copper-Catalyzed Ullmann Condensation : N-Arylation of Heterocyclic Compounds Containing an -NHCO- Moiety

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概要

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• N-Aryl heterocyclic compounds were synthesized from aryl halides and heterocyclic compounds containing an -NHCO- moiety by using a catalytic amount (1-10 mol%) of a commercially available copper catalyst in satisfactory yields. This catalytic reaction was applicable to the synthesis of N-aryl-2-pyridone, -2-pyrrolidone, -1(2H)-isoquinolone, -1(2H)-phthalazinone, -4(3H)-quinazolinone and -1,2,3-benzotriazin-4(3H)-one derivatives.

• 公益社団法人日本薬学会の論文
• 1997-04-15

著者

• Ukita Tatsuzo

  Lead Optimization Research Laboratory Tanabe Seiyaku Co. Ltd.

• SUGHARA Masakatsu

  Lead Optimization Research Laboratory, Tanabe Seiyaku Co., Ltd.,

• Sugahara M

  Tanabe Seiyaku Co. Ltd. Osaka Jpn

• Sugahara Masakatsu

  Lead Optimization Research Laboratory, Tanabe Seiyaku Co., Ltd.,

関連論文

• A Facile Copper-Catalyzed Ullmann Condensation : N-Arylation of Heterocyclic Compounds Containing an -NHCO- Moiety

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